Assay Detail
Binding
CHEMBL5626249
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Kv1.2 (unknown origin) expressed in Xenopus laevis Oocyte cells by electrophysiological recording
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | Oocyte |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Potassium voltage-gated channel subfamily A member 2 (CHEMBL2086) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Immunosuppressive effects of new thiophene-based K<sub>V</sub>1.3 inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.51 | 6.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5631442 | — | — | 1 | 6.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5631442 | — | IC50 | = | 308.0 | nM | 6.51 |