Assay Detail
Functional
CHEMBL5628812
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Antiproliferative activity against human MV4-11 cells assessed as reduction in cell viability after 72 hrs by CellTiterGlo assay
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MV4-11 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Rational discovery of dual FLT3/HDAC inhibitors as a potential AML therapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 6.01 | 8.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4077071 | — | — | 1 | 8.15 |
| CHEMBL5618643 | — | — | 1 | 7.04 |
| CHEMBL5632592 | — | — | 1 | 6.80 |
| CHEMBL5632493 | — | — | 1 | 6.43 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.38 |
| CHEMBL5631737 | — | — | 1 | 6.31 |
| CHEMBL5632450 | — | — | 1 | 6.16 |
| CHEMBL5631238 | — | — | 1 | 6.03 |
| CHEMBL5632762 | — | — | 1 | 6.00 |
| CHEMBL5631242 | — | — | 1 | 5.97 |
| CHEMBL5633405 | — | — | 1 | 5.80 |
| CHEMBL5633679 | — | — | 1 | 5.73 |
| CHEMBL5631257 | — | — | 1 | 5.69 |
| CHEMBL5633325 | — | — | 1 | 5.68 |
| CHEMBL5631818 | — | — | 1 | 5.43 |
| CHEMBL5633767 | — | — | 1 | 5.36 |
| CHEMBL5631871 | — | — | 1 | 5.32 |
| CHEMBL5632212 | — | — | 1 | 5.30 |
| CHEMBL5632335 | — | — | 1 | 5.28 |
| CHEMBL5633912 | — | — | 1 | 5.25 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4077071 | — | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL5618643 | — | IC50 | = | 92.0 | nM | 7.04 |
| CHEMBL5632592 | — | IC50 | = | 157.0 | nM | 6.80 |
| CHEMBL5632493 | — | IC50 | = | 367.0 | nM | 6.43 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 421.0 | nM | 6.38 |
| CHEMBL5631737 | — | IC50 | = | 487.0 | nM | 6.31 |
| CHEMBL5632450 | — | IC50 | = | 698.0 | nM | 6.16 |
| CHEMBL5631238 | — | IC50 | = | 934.0 | nM | 6.03 |
| CHEMBL5632762 | — | IC50 | = | 989.0 | nM | 6.00 |
| CHEMBL5631242 | — | IC50 | = | 1081.0 | nM | 5.97 |
| CHEMBL5633405 | — | IC50 | = | 1570.0 | nM | 5.80 |
| CHEMBL5633679 | — | IC50 | = | 1860.0 | nM | 5.73 |
| CHEMBL5631257 | — | IC50 | = | 2039.0 | nM | 5.69 |
| CHEMBL5633325 | — | IC50 | = | 2076.0 | nM | 5.68 |
| CHEMBL5631818 | — | IC50 | = | 3713.0 | nM | 5.43 |
| CHEMBL5633767 | — | IC50 | = | 4383.0 | nM | 5.36 |
| CHEMBL5631871 | — | IC50 | = | 4800.0 | nM | 5.32 |
| CHEMBL5632212 | — | IC50 | = | 4996.0 | nM | 5.30 |
| CHEMBL5632335 | — | IC50 | = | 5228.0 | nM | 5.28 |
| CHEMBL5633912 | — | IC50 | = | 5692.0 | nM | 5.25 |