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Assay Detail

CHEMBL5629550

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Toxicity
Cytotoxicity against human MRC5 cells assessed as reduction in cell viability incubated for 48 hrs by MTT assay
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Toxicity
Organism Homo sapiens
Cell Type MRC5
Confidence 1 — Organism
Curated By Autocuration

Target

MRC5 (CHEMBL614181)
Type CELL-LINE
Organism Homo sapiens

Publication

Cytotoxic effects of kinetin riboside and its selected analogues on cancer cell lines.
Totoń E, Lisiak N, Romaniuk-Drapała A, Framski G, Wyszko E, Ostrowski T.
Bioorg Med Chem Lett (2024) 100 : 129628 -129628
PubMed 38280656 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 8 5.55 6.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5633381 1 6.00
CHEMBL406643 1 5.68
CHEMBL411066 KINETIN RIBOSIDE 1 5.60
CHEMBL5632198 1 4.93
CHEMBL5632256 1 -
CHEMBL5632167 1 -
CHEMBL5632437 1 -
CHEMBL5629964 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5633381 IC50 = 1000.0 nM 6.00
CHEMBL406643 IC50 = 2100.0 nM 5.68
CHEMBL411066 KINETIN RIBOSIDE IC50 = 2500.0 nM 5.60
CHEMBL5632198 IC50 = 11700.0 nM 4.93
CHEMBL5632256 IC50 > 100000.0 nM -
CHEMBL5632167 IC50 > 100000.0 nM -
CHEMBL5632437 IC50 > 100000.0 nM -
CHEMBL5629964 IC50 > 100000.0 nM -