Assay Detail
Functional
CHEMBL5635763
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Cytotoxicity against human PANC-1 cells assessed as inhibition of cell growth measured after 72 hrs by Celltiter-Glo assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | PANC-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Recent advances in small molecule and peptide inhibitors of glucose-regulated protein 78 for cancer therapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.35 | 5.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1439833 | — | — | 1 | 5.35 |
| CHEMBL5647335 | — | — | 1 | - |
| CHEMBL5646586 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1439833 | — | IC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL5647335 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL5646586 | — | IC50 | > | 30000.0 | nM | - |