Assay Detail
Binding
CHEMBL5720962
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of PIK3C2A (unknown origin) by drug competition for substrate binding based assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha (CHEMBL1075102) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Inhibition of Human Class I vs Class III Phosphatidylinositol 3'-Kinases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 7.15 | 7.55 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1765602 | — | — | 1 | 7.55 |
| CHEMBL5723005 | — | — | 1 | 6.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1765602 | — | EC50 | = | 28.1 | nM | 7.55 |
| CHEMBL5723005 | — | EC50 | = | 176.0 | nM | 6.75 |