Assay Detail
Binding
CHEMBL5731069
Review assay metadata, readout intent, target linkage, and publication context from the same page.
TBD: TBD
21
Total Activities
7
Compounds Tested
3
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Protein tyrosine kinase modulators and methods of use
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 7.87 | 8.06 |
| kon | 7 | - | - |
| k_off | 7 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL6013504 | — | — | 3 | 8.06 |
| CHEMBL5951162 | — | — | 3 | 8.03 |
| CHEMBL5857101 | — | — | 3 | 7.96 |
| CHEMBL5871879 | — | — | 3 | 7.92 |
| CHEMBL5964556 | — | — | 3 | 7.82 |
| CHEMBL5847006 | — | — | 3 | 7.77 |
| CHEMBL5903567 | — | — | 3 | 7.55 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL6013504 | — | IC50 | = | 8.62 | nM | 8.06 |
| CHEMBL5951162 | — | IC50 | = | 9.33 | nM | 8.03 |
| CHEMBL5857101 | — | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL5871879 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL5964556 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL5847006 | — | IC50 | = | 17.0 | nM | 7.77 |
| CHEMBL5903567 | — | IC50 | = | 28.0 | nM | 7.55 |
| CHEMBL5903567 | — | kon | = | - | — | - |
| CHEMBL5903567 | — | k_off | = | - | s-1 | - |
| CHEMBL5871879 | — | kon | = | - | — | - |
| CHEMBL5871879 | — | k_off | = | - | s-1 | - |
| CHEMBL5847006 | — | kon | = | - | — | - |
| CHEMBL5847006 | — | k_off | = | - | s-1 | - |
| CHEMBL5951162 | — | k_off | = | - | s-1 | - |
| CHEMBL5964556 | — | kon | = | - | — | - |
| CHEMBL5964556 | — | k_off | = | - | s-1 | - |
| CHEMBL6013504 | — | kon | = | - | — | - |
| CHEMBL6013504 | — | k_off | = | - | s-1 | - |
| CHEMBL5857101 | — | kon | = | - | — | - |
| CHEMBL5857101 | — | k_off | = | - | s-1 | - |
| CHEMBL5951162 | — | kon | = | - | — | - |