Assay Detail
Binding
CHEMBL5732652
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition Assay: Inhibition of human tyrosine kinases.
39
Total Activities
13
Compounds Tested
3
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Compositions and methods for treating toxoplasmosis, cryptosporidiosis, and other apicomplexan protozoan related diseases
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 6.27 | 6.66 |
| kon | 13 | - | - |
| k_off | 13 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1785021 | — | — | 3 | 6.66 |
| CHEMBL2079214 | — | — | 3 | 6.61 |
| CHEMBL1785020 | — | — | 3 | 6.43 |
| CHEMBL2079138 | — | — | 3 | 6.27 |
| CHEMBL1231370 | — | — | 3 | 5.86 |
| CHEMBL2079168 | — | — | 3 | 5.79 |
| CHEMBL1231372 | — | — | 3 | - |
| CHEMBL2030553 | — | — | 3 | - |
| CHEMBL2030554 | — | — | 3 | - |
| CHEMBL2078800 | — | — | 3 | - |
| CHEMBL2079231 | — | — | 3 | - |
| CHEMBL2079139 | — | — | 3 | - |
| CHEMBL2079230 | — | — | 3 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1785021 | — | IC50 | = | 218.0 | nM | 6.66 |
| CHEMBL2079214 | — | IC50 | = | 244.0 | nM | 6.61 |
| CHEMBL1785020 | — | IC50 | = | 375.0 | nM | 6.43 |
| CHEMBL2079138 | — | IC50 | = | 541.0 | nM | 6.27 |
| CHEMBL1231370 | — | IC50 | = | 1382.0 | nM | 5.86 |
| CHEMBL2079168 | — | IC50 | = | 1613.0 | nM | 5.79 |
| CHEMBL1231370 | — | kon | = | - | — | - |
| CHEMBL2030554 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1231370 | — | k_off | = | - | s-1 | - |
| CHEMBL1231372 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1231372 | — | kon | = | - | — | - |
| CHEMBL1231372 | — | k_off | = | - | s-1 | - |
| CHEMBL1785020 | — | kon | = | - | — | - |
| CHEMBL1785020 | — | k_off | = | - | s-1 | - |
| CHEMBL1785021 | — | kon | = | - | — | - |
| CHEMBL2030554 | — | kon | = | - | — | - |
| CHEMBL2079138 | — | kon | = | - | — | - |
| CHEMBL2079138 | — | k_off | = | - | s-1 | - |
| CHEMBL2079214 | — | kon | = | - | — | - |
| CHEMBL2079214 | — | k_off | = | - | s-1 | - |
| CHEMBL2030553 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2030553 | — | k_off | = | - | s-1 | - |
| CHEMBL2079168 | — | kon | = | - | — | - |
| CHEMBL2030554 | — | k_off | = | - | s-1 | - |
| CHEMBL2030553 | — | kon | = | - | — | - |
| CHEMBL2078800 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2078800 | — | kon | = | - | — | - |
| CHEMBL2078800 | — | k_off | = | - | s-1 | - |
| CHEMBL2079231 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2079231 | — | kon | = | - | — | - |
| CHEMBL2079231 | — | k_off | = | - | s-1 | - |
| CHEMBL1785021 | — | k_off | = | - | s-1 | - |
| CHEMBL2079168 | — | k_off | = | - | s-1 | - |
| CHEMBL2079139 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2079139 | — | kon | = | - | — | - |
| CHEMBL2079139 | — | k_off | = | - | s-1 | - |
| CHEMBL2079230 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2079230 | — | kon | = | - | — | - |
| CHEMBL2079230 | — | k_off | = | - | s-1 | - |