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Assay Detail

CHEMBL615276

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Hepatitis B virus in 2.2.15 cell line
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HepG2
Confidence 1 — Organism
Curated By Intermediate

Target

HepG2 (CHEMBL395)
Type CELL-LINE
Organism Homo sapiens

Publication

Anti-human immunodeficiency and anti-hepatitis B virus activities of -l-2,3-dideoxy purine nucleosides
Bolon PJ, Peiyuan Wang, Chu CK, Gosselin G, Boudou V, Pierra C, Mathe C, Imbach J, Faraj A, Alaoui Ae, Sommadossi J, Pai S, Yong-Lian Zhu, Ju-Sheng Lin, Yung-Chi Cheng, Schinazi RF
Bioorg Med Chem Lett (1996) 6 : 1657 -1662
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 6 5.57 5.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL290427 1 5.92
CHEMBL23094 1 5.22
CHEMBL78101 1 -
CHEMBL45254 1 -
CHEMBL45071 1 -
CHEMBL1460 DIDANOSINE 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL290427 EC50 = 1200.0 nM 5.92
CHEMBL23094 EC50 = 6000.0 nM 5.22
CHEMBL78101 EC50 > 10000.0 nM -
CHEMBL45254 EC50 > 10000.0 nM -
CHEMBL45071 EC50 > 10000.0 nM -
CHEMBL1460 DIDANOSINE EC50 > 10000.0 nM -