Assay Detail
Functional
CHEMBL615641
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Compound was tested for the inhibitory activity of compound towards human rhinovirus 3C protease
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Enterovirus |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Design, synthesis, and evaluation of nonpeptidic inhibitors of human rhinovirus 3C protease.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 7.98 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL149950 | — | — | 1 | 8.70 |
| CHEMBL150011 | — | — | 1 | 7.96 |
| CHEMBL148483 | — | — | 1 | 7.29 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL149950 | — | Ki | = | 2.0 | nM | 8.70 |
| CHEMBL150011 | — | Ki | = | 11.0 | nM | 7.96 |
| CHEMBL148483 | — | Ki | = | 51.0 | nM | 7.29 |