Assay Detail
Binding
CHEMBL617189
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vivo binding affinity was evaluated against 5-hydroxytryptamine 2 receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Isoindolinone enantiomers having affinity for the dopamine D4 receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.64 | 7.84 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL37170 | — | — | 1 | 7.84 |
| CHEMBL35093 | — | — | 1 | 7.44 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL37170 | — | Ki | = | 14.6 | nM | 7.84 |
| CHEMBL35093 | — | Ki | = | 36.4 | nM | 7.44 |