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Assay Detail

CHEMBL617347

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound was evaluated for its binding against 5-hydroxytryptamine 2A receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

5-hydroxytryptamine receptor 2A (CHEMBL224)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Multistep solution-phase parallel synthesis of spiperone analogues.
Hansen HC, Olsson R, Croston G, Andersson CM.
Bioorg Med Chem Lett (2000) 10 : 2435 -2439
PubMed 11078195 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.70 7.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL81377 1 7.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL81377 Ki = 20.0 nM 7.70