Assay Detail
Binding
CHEMBL618079
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Binding affinity towards murine 5-hydroxytryptamine 5A receptor
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 5.67 | 6.67 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL266250 | — | — | 1 | 6.67 |
| CHEMBL92879 | — | — | 1 | 5.28 |
| CHEMBL478 | CHLOROPHENYLPIPERAZINE | 2.0 | 1 | 5.06 |
| CHEMBL18772 | QUIPAZINE | 2.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL266250 | — | Ki | = | 215.0 | nM | 6.67 |
| CHEMBL92879 | — | Ki | = | 5300.0 | nM | 5.28 |
| CHEMBL478 | CHLOROPHENYLPIPERAZINE | Ki | = | 8700.0 | nM | 5.06 |
| CHEMBL18772 | QUIPAZINE | Ki | > | 10000.0 | nM | - |