Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL619009

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound was tested for its binding affinity for 5-hydroxytryptamine 4 receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

5-hydroxytryptamine receptor 4 (CHEMBL1875)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

SB-656104-A: a novel 5-HT(7) receptor antagonist with improved in vivo properties.
Forbes IT, Douglas S, Gribble AD, Ife RJ, Lightfoot AP, Garner AE, Riley GJ, Jeffrey P, Stevens AJ, Stean TO, Thomas DR.
Bioorg Med Chem Lett (2002) 12 : 3341 -3344
PubMed 12392747 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.72 5.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL95104 1 5.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL95104 Ki = 1905.46 nM 5.72