Assay Detail
Functional
CHEMBL620609
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Tested for 5-hydroxytryptamine 4 receptor antagonist activity
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
5-HT4 receptor ligands: applications and new prospects.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.61 | 8.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL97019 | — | — | 1 | 8.17 |
| CHEMBL99591 | — | — | 1 | 7.04 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL97019 | — | Ki | = | 6.7 | nM | 8.17 |
| CHEMBL99591 | — | Ki | = | 91.9 | nM | 7.04 |