Assay Detail

CHEMBL629640

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Physicochemical

Dissociation constant of the compound; value ranges from 0.81-1.2 nM

ChEMBL ↗

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Target

No relevant target (CHEMBL2362975) ↗

Open DB target context

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No relevant target (CHEMBL2362975) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target No relevant target

CHEMBL2362975

Anchored from Assay target.

Protein identity No relevant target

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Physicochemical
Confidence	0 — Uncurated / Unknown
Curated By	Autocuration

Target

No relevant target (CHEMBL2362975) ↗

Type

NO TARGET

Publication

N-fluoroalkylated and N-alkylated analogues of the dopaminergic D-2 receptor antagonist raclopride.

Lannoye GS, Moerlein SM, Parkinson D, Welch MJ.
J Med Chem (1990) 33 : 2430 -2437
PubMed 2391685 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
Kd	1	9.09	9.09

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL8809	RACLOPRIDE	2.0	1	9.09

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL8809	RACLOPRIDE	Kd	=	0.81	nM	9.09