Assay Detail
Physicochemical
CHEMBL630131
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Dissociation constant was reported
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Physicochemical |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Inhibition of dopamine receptors by endogenous amines: binding to striatal receptors and pharmacological effects on locomotor activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 8.96 | 9.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL44877 | — | — | 1 | 9.70 |
| CHEMBL21640 | — | — | 1 | 8.89 |
| CHEMBL298285 | — | — | 1 | 8.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL44877 | — | Kd | = | 0.2 | nM | 9.70 |
| CHEMBL21640 | — | Kd | = | 1.3 | nM | 8.89 |
| CHEMBL298285 | — | Kd | = | 5.0 | nM | 8.30 |