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Assay Detail

CHEMBL638726

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity for adenosine A1 receptor using [3H]- CHA or [3H]- PIA in bovine brain cortical membranes
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Bos taurus
Confidence 9 — Direct single protein target
Curated By Expert

Target

Adenosine receptor A1 (CHEMBL4975)
Type SINGLE PROTEIN
Organism Bos taurus

Publication

Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.
Jacobson KA, van Galen PJ, Williams M.
J Med Chem (1992) 35 : 407 -422
PubMed 1738138 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 10.00 10.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL133982 1 10.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL133982 Ki = 0.1 nM 10.00