Assay Detail
Binding
CHEMBL640603
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity for Adenosine A1 receptor using [125I]-ABA in chick cerebellar membrane
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Tissue | Cerebellum |
| Subcellular | Membrane |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
N6-phenyladenosines: pronounced effect of phenyl substituents on affinity for A2 adenosine receptors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.96 | 7.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL609650 | — | — | 1 | 7.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL609650 | — | IC50 | = | 11.1 | nM | 7.96 |