Assay Detail
Binding
CHEMBL640606
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity against bovine brain adenosine A1 receptor using N6-[3H]- cyclohexyladenosine
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Synthesis of xanthines as adenosine antagonists, a practical quantitative structure-activity relationship application.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.61 | 5.61 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1355736 | THEOPHYLLINE | 4.0 | 1 | 5.61 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1355736 | THEOPHYLLINE | IC50 | = | 2430.0 | nM | 5.61 |