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Assay Detail

CHEMBL640612

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity of [3H]-MRE 2029-F20 towards human adenosine A2b receptor expressed in CHO cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type CHO
Confidence 9 — Direct single protein target
Curated By Expert

Target

Adenosine receptor A2b (CHEMBL255)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

A mild, efficient and alpha-selective glycosidation by using potassium dodecatungstocobaltate trihydrate as catalyst.
Rafiee E, Tangestaninejad S, Habibi MH, Mirkhani V.
Bioorg Med Chem Lett (2004) 14 : 3611 -3614
PubMed 15177485 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 8.78 8.78

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL260331 1 8.78

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL260331 Kd = 1.65 nM 8.78