Assay Detail
Binding
CHEMBL644359
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity towards Alpha-2 adrenergic receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.38 | 7.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL92221 | — | — | 1 | 7.72 |
| CHEMBL27251 | — | — | 1 | 7.03 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL92221 | — | Ki | = | 19.0 | nM | 7.72 |
| CHEMBL27251 | — | Ki | = | 92.8 | nM | 7.03 |