Assay Detail
Binding
CHEMBL644595
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of aminopeptidase M or membrane leucine aminopeptidase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Inhibition of aminopeptidases by peptides containing ketomethylene and hydroxyethylene amide bond replacements.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.53 | 7.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL28650 | AMASTATIN | — | 1 | 7.70 |
| CHEMBL29292 | UBENIMEX | 2.0 | 1 | 5.36 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL28650 | AMASTATIN | Ki | = | 20.0 | nM | 7.70 |
| CHEMBL29292 | UBENIMEX | Ki | = | 4400.0 | nM | 5.36 |