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Assay Detail

CHEMBL646998

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity at alpha 2B adrenergic receptor of rat.
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Alpha-2B adrenergic receptor (CHEMBL266)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Binding of beta-carbolines at imidazoline I2 receptors: a structure-affinity investigation.
Glennon RA, Grella B, Tyacke RJ, Lau A, Westaway J, Hudson AL.
Bioorg Med Chem Lett (2004) 14 : 999 -1002
PubMed 15013009 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 6.85 6.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL6310 1 6.85

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL6310 Ki = 140.0 nM 6.85