Assay Detail
Binding
CHEMBL647121
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Inhibition constant against Angiotensin II receptor, type 1 was determined
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Angiotensin II AT1 receptor antagonists. Clinical implications of active metabolites.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.88 | 6.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL74767 | — | — | 1 | 6.43 |
| CHEMBL1069 | VALSARTAN | 4.0 | 1 | 5.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL74767 | — | Ki | = | 370.0 | nM | 6.43 |
| CHEMBL1069 | VALSARTAN | Ki | = | 4700.0 | nM | 5.33 |