Assay Detail
Binding
CHEMBL648565
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Tested for binding affinity to Angiotensin II receptor, type 1
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
A potent long-acting imidazole-5-acrylic acid angiotensin II AT-1 receptor antagonist
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.85 | 6.36 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL55508 | — | — | 1 | 6.36 |
| CHEMBL289543 | — | — | 1 | 5.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL55508 | — | IC50 | = | 440.0 | nM | 6.36 |
| CHEMBL289543 | — | IC50 | = | 4530.0 | nM | 5.34 |