Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL648648

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
In vitro binding affinity for PBR (peripheral benzodiazepine receptor) in monkey brain
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Translocator protein (CHEMBL5742)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

[18F]FMDAA1106 and [18F]FEDAA1106: two positron-emitter labeled ligands for peripheral benzodiazepine receptor (PBR).
Zhang MR, Maeda J, Furutsuka K, Yoshida Y, Ogawa M, Suhara T, Suzuki K.
Bioorg Med Chem Lett (2003) 13 : 201 -204
PubMed 12482423 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 9.73 9.73

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL63064 1 9.73

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL63064 Ki = 0.188 nM 9.73