Assay Detail
Binding
CHEMBL648740
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Ancillary Binding affinity towards rat alpha-2B receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Two novel and potent 3-[(o-methoxyphenyl)piperazinylethyl]-5-phenylthien.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.17 | 7.18 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL13856 | A-123189 | — | 1 | 7.18 |
| CHEMBL268758 | A-119637 | — | 1 | 7.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL13856 | A-123189 | Ki | = | 66.6 | nM | 7.18 |
| CHEMBL268758 | A-119637 | Ki | = | 71.0 | nM | 7.15 |