Assay Detail
Binding
CHEMBL650008
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Binding affinity against aspartic protease renin.
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Protease inhibitors: current status and future prospects.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 8.72 | 9.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL31601 | REMIKIREN | 2.0 | 1 | 9.15 |
| CHEMBL293196 | — | — | 1 | 9.15 |
| CHEMBL323839 | — | — | 1 | 7.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL31601 | REMIKIREN | Ki | = | 0.7 | nM | 9.15 |
| CHEMBL293196 | — | Ki | = | 0.7 | nM | 9.15 |
| CHEMBL323839 | — | Ki | = | 14.0 | nM | 7.85 |