Assay Detail
Binding
CHEMBL652863
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Tested for binding affinity against angiotensin II receptor in rat adrenal cortex
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Tissue | Adrenal cortex |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Uracil-based angiotensin II receptor antagonists
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.11 | 8.36 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL305032 | — | — | 1 | 8.36 |
| CHEMBL62314 | — | — | 1 | 7.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL305032 | — | IC50 | = | 4.4 | nM | 8.36 |
| CHEMBL62314 | — | IC50 | = | 14.0 | nM | 7.85 |