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Assay Detail

CHEMBL653009

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound was tested for its binding affinity against mouse spleen Cannabinoid receptor 2 using [3H]CP-55940 as radioligand
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Tissue Spleen
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Cannabinoid receptor 2 (CHEMBL5373)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Pharmacophoric requirements for the cannabinoid side chain. Probing the cannabinoid receptor subsite at C1'.
Papahatjis DP, Nikas SP, Kourouli T, Chari R, Xu W, Pertwee RG, Makriyannis A.
J Med Chem (2003) 46 : 3221 -3229
PubMed 12852753 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 9.66 9.66

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL108085 1 9.66

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL108085 Ki = 0.22 nM 9.66