Assay Detail
Binding
CHEMBL653246
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Inhibitor concentration against Beta-galactosidase from Aspergillus niger
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Aspergillus niger |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
Synthesis of [(2S,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]-5-methylfuran-4-carboxylic acid derivatives: new leads as selective beta-galactosidase inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.84 | 5.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2114148 | — | — | 1 | 5.12 |
| CHEMBL2114149 | — | — | 1 | 4.55 |
| CHEMBL3350284 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2114148 | — | IC50 | = | 7500.0 | nM | 5.12 |
| CHEMBL2114149 | — | IC50 | = | 28000.0 | nM | 4.55 |
| CHEMBL3350284 | — | IC50 | = | 370000.0 | nM | - |