Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL653508

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibitory activity against recombinant human Beta-secretase 1
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Beta-secretase 1 (CHEMBL4822)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Green tea catechins as a BACE1 (beta-secretase) inhibitor.
Jeon SY, Bae K, Seong YH, Song KS.
Bioorg Med Chem Lett (2003) 13 : 3905 -3908
PubMed 14592472 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 3 6.24 6.77

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL126079 1 6.77
CHEMBL338988 1 6.68
CHEMBL126142 1 5.28

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL126079 Ki = 170.0 nM 6.77
CHEMBL338988 Ki = 210.0 nM 6.68
CHEMBL126142 Ki = 5300.0 nM 5.28