Assay Detail
Binding
CHEMBL654865
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Compound was evaluated for the protection of butyrylcholinesterase against DFT in mice and expressed as Ki
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
N-allyl analogues of phencyclidine: chemical synthesis and pharmacological properties.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 5.48 | 6.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL23626 | — | — | 1 | 6.30 |
| CHEMBL23627 | — | — | 1 | 5.58 |
| CHEMBL281855 | — | — | 1 | 4.57 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL23626 | — | Ki | = | 500.0 | nM | 6.30 |
| CHEMBL23627 | — | Ki | = | 2600.0 | nM | 5.58 |
| CHEMBL281855 | — | Ki | = | 27000.0 | nM | 4.57 |