Assay Detail
Binding
CHEMBL655438
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The compound was tested for the inhibition of Carboxypeptidase A
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
2-Benzyl-3,4-iminobutanoic acid as inhibitor of carboxypeptidase A.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 8 | 5.28 | 6.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL33352 | — | — | 1 | 6.10 |
| CHEMBL321983 | — | — | 1 | 4.46 |
| CHEMBL318559 | — | — | 1 | - |
| CHEMBL318266 | — | — | 1 | - |
| CHEMBL320875 | — | — | 1 | - |
| CHEMBL100123 | — | — | 1 | - |
| CHEMBL101276 | — | — | 1 | - |
| CHEMBL100122 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL33352 | — | Ki | = | 800.0 | nM | 6.10 |
| CHEMBL321983 | — | Ki | = | 35000.0 | nM | 4.46 |
| CHEMBL318559 | — | Ki | = | 510000.0 | nM | - |
| CHEMBL318266 | — | Ki | = | 120000.0 | nM | - |
| CHEMBL320875 | — | Ki | = | 803000.0 | nM | - |
| CHEMBL100123 | — | Ki | = | 792000.0 | nM | - |
| CHEMBL101276 | — | Ki | = | 646000.0 | nM | - |
| CHEMBL100122 | — | Ki | = | 230000.0 | nM | - |