Assay Detail
Binding
CHEMBL655812
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition against CD23 (IgE receptor) proteolysis in membranes derived from RPM18866 cells
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Target
Low affinity immunoglobulin epsilon Fc receptor (CHEMBL2940) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Selective inhibition of low affinity IgE receptor (CD23) processing.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 22 | 6.83 | 7.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL115348 | — | — | 1 | 7.92 |
| CHEMBL118054 | — | — | 1 | 7.89 |
| CHEMBL324564 | — | — | 1 | 7.80 |
| CHEMBL115326 | — | — | 1 | 7.70 |
| CHEMBL424251 | — | — | 1 | 7.52 |
| CHEMBL326148 | — | — | 1 | 7.22 |
| CHEMBL116506 | — | — | 1 | 7.10 |
| CHEMBL116435 | — | — | 1 | 7.00 |
| CHEMBL320798 | — | — | 1 | 7.00 |
| CHEMBL279786 | BATIMASTAT | 2.0 | 1 | 7.00 |
| CHEMBL326814 | — | — | 1 | 6.89 |
| CHEMBL114332 | — | — | 1 | 6.89 |
| CHEMBL324723 | — | — | 1 | 6.89 |
| CHEMBL113764 | — | — | 1 | 6.80 |
| CHEMBL325608 | — | — | 1 | 6.68 |
| CHEMBL433197 | — | — | 1 | 6.42 |
| CHEMBL96654 | — | — | 1 | 5.72 |
| CHEMBL326985 | — | — | 1 | 5.52 |
| CHEMBL112228 | — | — | 1 | 5.43 |
| CHEMBL94155 | — | — | 1 | 5.30 |
| CHEMBL324295 | — | — | 1 | - |
| CHEMBL117823 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL115348 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL118054 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL324564 | — | IC50 | = | 16.0 | nM | 7.80 |
| CHEMBL115326 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL424251 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL326148 | — | IC50 | = | 60.0 | nM | 7.22 |
| CHEMBL116506 | — | IC50 | = | 80.0 | nM | 7.10 |
| CHEMBL116435 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL320798 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL279786 | BATIMASTAT | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL326814 | — | IC50 | = | 130.0 | nM | 6.89 |
| CHEMBL114332 | — | IC50 | = | 130.0 | nM | 6.89 |
| CHEMBL324723 | — | IC50 | = | 130.0 | nM | 6.89 |
| CHEMBL113764 | — | IC50 | = | 160.0 | nM | 6.80 |
| CHEMBL325608 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL433197 | — | IC50 | = | 380.0 | nM | 6.42 |
| CHEMBL96654 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL326985 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL112228 | — | IC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL94155 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL324295 | — | IC50 | ~ | 100.0 | nM | - |
| CHEMBL117823 | — | IC50 | ~ | 1000.0 | nM | - |