Assay Detail
Functional
CHEMBL655889
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.
37
Total Activities
37
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | CHO |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Design of selective peptidomimetic agonists for the human orphan receptor BRS-3.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 37 | 7.30 | 9.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL57104 | — | — | 1 | 9.72 |
| CHEMBL56369 | — | — | 1 | 8.85 |
| CHEMBL57438 | — | — | 1 | 8.82 |
| CHEMBL3144501 | — | — | 1 | 8.68 |
| CHEMBL294647 | — | — | 1 | 8.66 |
| CHEMBL57039 | — | — | 1 | 8.54 |
| CHEMBL57559 | — | — | 1 | 8.51 |
| CHEMBL3144492 | — | — | 1 | 8.40 |
| CHEMBL56626 | — | — | 1 | 8.22 |
| CHEMBL3144493 | — | — | 1 | 8.11 |
| CHEMBL292646 | — | — | 1 | 8.03 |
| CHEMBL56562 | — | — | 1 | 7.82 |
| CHEMBL57068 | — | — | 1 | 7.77 |
| CHEMBL175651 | — | — | 1 | 7.72 |
| CHEMBL292176 | — | — | 1 | 7.68 |
| CHEMBL417767 | — | — | 1 | 7.68 |
| CHEMBL418147 | — | — | 1 | 7.62 |
| CHEMBL3144491 | — | — | 1 | 7.60 |
| CHEMBL60537 | — | — | 1 | 7.52 |
| CHEMBL3144500 | — | — | 1 | 7.50 |
| CHEMBL3144495 | — | — | 1 | 7.34 |
| CHEMBL3144499 | — | — | 1 | 7.24 |
| CHEMBL293820 | — | — | 1 | 7.16 |
| CHEMBL3144490 | — | — | 1 | 7.10 |
| CHEMBL3144489 | — | — | 1 | 6.85 |
| CHEMBL262992 | — | — | 1 | 6.82 |
| CHEMBL3144502 | — | — | 1 | 6.64 |
| CHEMBL5483013 | — | — | 1 | 6.62 |
| CHEMBL3144496 | — | — | 1 | 6.51 |
| CHEMBL3144497 | — | — | 1 | 6.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL57104 | — | EC50 | = | 0.19 | nM | 9.72 |
| CHEMBL56369 | — | EC50 | = | 1.4 | nM | 8.85 |
| CHEMBL57438 | — | EC50 | = | 1.5 | nM | 8.82 |
| CHEMBL3144501 | — | EC50 | = | 2.1 | nM | 8.68 |
| CHEMBL294647 | — | EC50 | = | 2.2 | nM | 8.66 |
| CHEMBL57039 | — | EC50 | = | 2.9 | nM | 8.54 |
| CHEMBL57559 | — | EC50 | = | 3.1 | nM | 8.51 |
| CHEMBL3144492 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL56626 | — | EC50 | = | 6.0 | nM | 8.22 |
| CHEMBL3144493 | — | EC50 | = | 7.8 | nM | 8.11 |
| CHEMBL292646 | — | EC50 | = | 9.3 | nM | 8.03 |
| CHEMBL56562 | — | EC50 | = | 15.0 | nM | 7.82 |
| CHEMBL57068 | — | EC50 | = | 17.0 | nM | 7.77 |
| CHEMBL175651 | — | EC50 | = | 19.0 | nM | 7.72 |
| CHEMBL417767 | — | EC50 | = | 21.0 | nM | 7.68 |
| CHEMBL292176 | — | EC50 | = | 21.0 | nM | 7.68 |
| CHEMBL418147 | — | EC50 | = | 24.0 | nM | 7.62 |
| CHEMBL3144491 | — | EC50 | = | 25.0 | nM | 7.60 |
| CHEMBL60537 | — | EC50 | = | 30.0 | nM | 7.52 |
| CHEMBL3144500 | — | EC50 | = | 32.0 | nM | 7.50 |
| CHEMBL3144495 | — | EC50 | = | 46.0 | nM | 7.34 |
| CHEMBL3144499 | — | EC50 | = | 57.0 | nM | 7.24 |
| CHEMBL293820 | — | EC50 | = | 70.0 | nM | 7.16 |
| CHEMBL3144490 | — | EC50 | = | 79.0 | nM | 7.10 |
| CHEMBL3144489 | — | EC50 | = | 140.0 | nM | 6.85 |
| CHEMBL262992 | — | EC50 | = | 151.0 | nM | 6.82 |
| CHEMBL3144502 | — | EC50 | = | 230.0 | nM | 6.64 |
| CHEMBL5483013 | — | EC50 | = | 240.0 | nM | 6.62 |
| CHEMBL3144496 | — | EC50 | = | 310.0 | nM | 6.51 |
| CHEMBL3144497 | — | EC50 | = | 710.0 | nM | 6.15 |
| CHEMBL3144503 | — | EC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL3144498 | — | EC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL57046 | — | EC50 | = | 2700.0 | nM | 5.57 |
| CHEMBL403317 | — | EC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL3144494 | — | EC50 | = | 6400.0 | nM | 5.19 |
| CHEMBL438926 | — | EC50 | = | 6400.0 | nM | 5.19 |
| CHEMBL58097 | — | EC50 | = | 7900.0 | nM | 5.10 |