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Assay Detail

CHEMBL655958

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity of compound against normal human ovarian C18013S cell line
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type C180-13S
Confidence 1 — Organism
Curated By Intermediate

Target

C180-13S (CHEMBL613540)
Type CELL-LINE
Organism Homo sapiens

Publication

Antiproliferative and phenotype-transforming antitumor agents derived from cysteine.
Glenn MP, Kahnberg P, Boyle GM, Hansford KA, Hans D, Martyn AC, Parsons PG, Fairlie DP.
J Med Chem (2004) 47 : 2984 -2994
PubMed 15163181 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 6.36 7.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL99 TRICHOSTATIN 1.0 1 7.22
CHEMBL101006 1 6.40
CHEMBL103508 1 6.22
CHEMBL318384 1 6.16
CHEMBL103379 1 5.82

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL99 TRICHOSTATIN IC50 = 60.0 nM 7.22
CHEMBL101006 IC50 = 400.0 nM 6.40
CHEMBL103508 IC50 = 600.0 nM 6.22
CHEMBL318384 IC50 = 700.0 nM 6.16
CHEMBL103379 IC50 = 1500.0 nM 5.82