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Assay Detail

CHEMBL656590

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
The compound was tested for cytotoxic activity against CH1 cell line(human ovarian carcinoma )
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type CH1
Confidence 1 — Organism
Curated By Intermediate

Target

CH1 (CHEMBL614455)
Type CELL-LINE
Organism Homo sapiens

Publication

N4-(omega-Aminoalkyl)-1-[(omega-aminoalkyl)amino]-4- acridinecarboxamides: novel, potent, cytotoxic, and DNA-binding agents.
Antonini I, Polucci P, Kelland LR, Spinelli S, Pescalli N, Martelli S.
J Med Chem (2000) 43 : 4801 -4805
PubMed 11123989 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 7.11 8.20

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL53463 DOXORUBICIN 4.0 1 8.20
CHEMBL342519 1 7.05
CHEMBL141654 1 6.07

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL53463 DOXORUBICIN IC50 = 6.3 nM 8.20
CHEMBL342519 IC50 = 89.0 nM 7.05
CHEMBL141654 IC50 = 860.0 nM 6.07