Assay Detail
Binding
CHEMBL657103
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Inhibitory concentration against Human pancreatic Chymotrypsin
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
P1 Phenethyl peptide boronic acid inhibitors of HCV NS3 protease.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 6 | 4.70 | 4.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL107287 | — | — | 1 | 4.70 |
| CHEMBL262398 | — | — | 1 | - |
| CHEMBL413150 | — | — | 1 | - |
| CHEMBL432959 | — | — | 1 | - |
| CHEMBL324207 | — | — | 1 | - |
| CHEMBL108657 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL107287 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL262398 | — | IC50 | > | 60000.0 | nM | - |
| CHEMBL413150 | — | IC50 | > | 60000.0 | nM | - |
| CHEMBL432959 | — | IC50 | > | 48000.0 | nM | - |
| CHEMBL324207 | — | IC50 | > | 60000.0 | nM | - |
| CHEMBL108657 | — | IC50 | > | 60000.0 | nM | - |