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Assay Detail

CHEMBL657193

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Binding
Inhibition of human carbonic anhydrase II
31
Total Activities
31
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Carbonic anhydrase 2 (CHEMBL205)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
Winum JY, Vullo D, Casini A, Montero JL, Scozzafava A, Supuran CT.
J Med Chem (2003) 46 : 2197 -2204
PubMed 12747791 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 31 7.74 8.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL23350 1 8.96
CHEMBL24259 PHENYLSULFAMATE 1 8.89
CHEMBL283121 1 8.82
CHEMBL23258 1 8.82
CHEMBL71872 1 8.80
CHEMBL24210 1 8.72
CHEMBL24261 OCTYL SULFAMATE 1 8.57
CHEMBL69948 1 8.54
CHEMBL24120 1 8.42
CHEMBL221802 1 8.30
CHEMBL220492 TOPIRAMATE 4.0 1 8.30
CHEMBL18 ETHOXZOLAMIDE 4.0 1 8.10
CHEMBL122708 EMATE 1 8.00
CHEMBL20 ACETAZOLAMIDE 4.0 1 7.92
CHEMBL220493 1 7.89
CHEMBL19 METHAZOLAMIDE 4.0 1 7.85
CHEMBL302593 1 7.82
CHEMBL68590 1 7.75
CHEMBL544763 1 7.64
CHEMBL71371 1 7.57
CHEMBL71549 1 7.54
CHEMBL67749 1 7.20
CHEMBL68257 1 7.12
CHEMBL417287 1 7.02
CHEMBL69322 1 7.01
CHEMBL68536 PERFLUOROPHENYL SULFAMATE 1 6.95
CHEMBL71873 SULFAMIC ACID PENTACHLOROPHENYL ESTER 1 6.90
CHEMBL303601 1 6.86
CHEMBL303942 1 6.86
CHEMBL24119 1 6.83

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL23350 Ki = 1.1 nM 8.96
CHEMBL24259 PHENYLSULFAMATE Ki = 1.3 nM 8.89
CHEMBL283121 Ki = 1.5 nM 8.82
CHEMBL23258 Ki = 1.5 nM 8.82
CHEMBL71872 Ki = 1.6 nM 8.80
CHEMBL24210 Ki = 1.9 nM 8.72
CHEMBL24261 OCTYL SULFAMATE Ki = 2.7 nM 8.57
CHEMBL69948 Ki = 2.9 nM 8.54
CHEMBL24120 Ki = 3.8 nM 8.42
CHEMBL221802 Ki = 5.0 nM 8.30
CHEMBL220492 TOPIRAMATE Ki = 5.0 nM 8.30
CHEMBL18 ETHOXZOLAMIDE Ki = 8.0 nM 8.10
CHEMBL122708 EMATE Ki = 10.0 nM 8.00
CHEMBL20 ACETAZOLAMIDE Ki = 12.0 nM 7.92
CHEMBL220493 Ki = 13.0 nM 7.89
CHEMBL19 METHAZOLAMIDE Ki = 14.0 nM 7.85
CHEMBL302593 Ki = 15.0 nM 7.82
CHEMBL68590 Ki = 18.0 nM 7.75
CHEMBL544763 Ki = 23.0 nM 7.64
CHEMBL71371 Ki = 27.0 nM 7.57
CHEMBL71549 Ki = 29.0 nM 7.54
CHEMBL67749 Ki = 63.0 nM 7.20
CHEMBL68257 Ki = 76.0 nM 7.12
CHEMBL417287 Ki = 95.0 nM 7.02
CHEMBL69322 Ki = 98.0 nM 7.01
CHEMBL68536 PERFLUOROPHENYL SULFAMATE Ki = 113.0 nM 6.95
CHEMBL71873 SULFAMIC ACID PENTACHLOROPHENYL ESTER Ki = 125.0 nM 6.90
CHEMBL303601 Ki = 138.0 nM 6.86
CHEMBL303942 Ki = 138.0 nM 6.86
CHEMBL24119 Ki = 149.0 nM 6.83
CHEMBL68253 SULFAMATE Ki = 97000.0 nM 4.01