Assay Detail

CHEMBL657379

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Functional

Antagonistic activity against cholecystokinin type A receptor

ChEMBL ↗

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Target

Cholecystokinin receptor type A (CHEMBL1901) ↗

Open DB target context

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Cholecystokinin receptor type A (CHEMBL1901) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target Cholecystokinin receptor type A

CHEMBL1901

Anchored from Assay target.

Protein identity Cholecystokinin receptor type A

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Functional
Confidence	8 — Homologous single protein target
Curated By	Autocuration

Target

Cholecystokinin receptor type A (CHEMBL1901) ↗

Type	SINGLE PROTEIN
Organism	Homo sapiens

Publication

Excursions in drug discovery.

Patchett AA.
J Med Chem (1993) 36 : 2051 -2058
PubMed 8340909 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	2	7.98	10.10

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL9506	DEVAZEPIDE	2.0	1	10.10
CHEMBL283117	ASPERLICIN	—	1	5.85

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL9506	DEVAZEPIDE	IC50	=	0.08	nM	10.10
CHEMBL283117	ASPERLICIN	IC50	=	1400.0	nM	5.85