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Assay Detail

CHEMBL657903

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity towards Cannabinoid receptor 1
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Cannabinoid receptor 1 (CHEMBL218)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Synthesis and testing of novel phenyl substituted side-chain analogues of classical cannabinoids.
Krishnamurthy M, Ferreira AM, Moore BM.
Bioorg Med Chem Lett (2003) 13 : 3487 -3490
PubMed 14505654 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.73 8.73

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL117033 1 8.73

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL117033 Ki = 1.86 nM 8.73