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Assay Detail

CHEMBL657913

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound was tested for inhibition of Adenylyl cyclase in cannabinoid receptor 1 (CB1).
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Cannabinoid receptor 1 (CHEMBL218)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Novel cannabinol probes for CB1 and CB2 cannabinoid receptors.
Mahadevan A, Siegel C, Martin BR, Abood ME, Beletskaya I, Razdan RK.
J Med Chem (2000) 43 : 3778 -3785
PubMed 11020293 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.70 8.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL109393 1 8.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL109393 Ki = 2.0 nM 8.70