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Assay Detail

CHEMBL657997

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity for the Cannabinoid receptor using [3H]CP-55940 as radioligand
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Cannabinoid receptor 1 (CHEMBL3571)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Enantioselective synthesis and pharmacology of 11-hydroxy-(1'S,2'R)-dimethylheptyl-delta 8-THC.
Liddle J, Huffman JW, Wiley JL, Martin BR.
Bioorg Med Chem Lett (1998) 8 : 2223 -2226
PubMed 9873517 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 9.14 9.14

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL307696 1 9.14

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL307696 Ki = 0.73 nM 9.14