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Assay Detail

CHEMBL658285

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of ovine CRF stimulated adenylate cyclase assay in CHO-p5 cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Ovis aries
Cell Type CHO-p5
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Corticotropin releasing factor (CRF) receptor modulators: progress and opportunities for new therapeutic agents.
Gilligan PJ, Robertson DW, Zaczek R.
J Med Chem (2000) 43 : 1641 -1660
PubMed 10794681 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.45 6.45

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL290762 1 6.45

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL290762 IC50 = 357.0 nM 6.45