Assay Detail
Binding
CHEMBL658970
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Compound was evaluated for its binding affinity for mouse spleen Cannabinoid receptor 2
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Tissue | Spleen |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Head group analogs of arachidonylethanolamide, the endogenous cannabinoid ligand.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 7 | 5.43 | 6.09 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL120526 | METHANANDAMIDE | — | 1 | 6.09 |
| CHEMBL15848 | ANANDAMIDE | — | 1 | 5.71 |
| CHEMBL137899 | — | — | 1 | 5.68 |
| CHEMBL141647 | — | — | 1 | 5.51 |
| CHEMBL342659 | — | — | 1 | 5.20 |
| CHEMBL434069 | — | — | 1 | 4.96 |
| CHEMBL39878 | — | — | 1 | 4.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL120526 | METHANANDAMIDE | Ki | = | 815.0 | nM | 6.09 |
| CHEMBL15848 | ANANDAMIDE | Ki | = | 1926.0 | nM | 5.71 |
| CHEMBL137899 | — | Ki | = | 2100.0 | nM | 5.68 |
| CHEMBL141647 | — | Ki | = | 3100.0 | nM | 5.51 |
| CHEMBL342659 | — | Ki | = | 6300.0 | nM | 5.20 |
| CHEMBL434069 | — | Ki | = | 11000.0 | nM | 4.96 |
| CHEMBL39878 | — | Ki | = | 13000.0 | nM | 4.89 |