Assay Detail
Binding
CHEMBL660636
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Compound was evaluated for its activity against bacterial DNA gyrase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bacteria |
| Confidence | 3 — Cell-line / Tissue |
| Curated By | Intermediate |
Publication
3-benzyl-quinolones: Novel, potent inhibitors of mammalian topoisomerase II
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 6.85 | 6.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL440642 | — | — | 1 | 6.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL440642 | — | EC50 | = | 140.0 | nM | 6.85 |