Assay Detail
Binding
CHEMBL661059
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity for the cannabinoid brain receptor (CB1) using [3H]CP-55940
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Enantioselective synthesis and pharmacology of 11-hydroxy-(1'S,2'R)-dimethylheptyl-delta 8-THC.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 9.25 | 9.34 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL71401 | — | — | 1 | 9.34 |
| CHEMBL73060 | — | — | 1 | 9.31 |
| CHEMBL411626 | — | — | 1 | 9.11 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL71401 | — | Ki | = | 0.46 | nM | 9.34 |
| CHEMBL73060 | — | Ki | = | 0.49 | nM | 9.31 |
| CHEMBL411626 | — | Ki | = | 0.77 | nM | 9.11 |