Assay Detail
Binding
CHEMBL661829
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Compound was evaluated for the binding affinity against CCK A receptor in cortical cells.
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
Hybrid cholecystokinin (CCK) antagonists: new implications in the design and modification of CCK antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 4.96 | 5.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL112222 | — | — | 1 | 5.89 |
| CHEMBL349857 | — | — | 1 | 4.96 |
| CHEMBL9485 | — | — | 1 | 4.91 |
| CHEMBL158362 | — | — | 1 | 4.72 |
| CHEMBL162111 | — | — | 1 | 4.32 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL112222 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL349857 | — | IC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL9485 | — | IC50 | = | 12400.0 | nM | 4.91 |
| CHEMBL158362 | — | IC50 | = | 19000.0 | nM | 4.72 |
| CHEMBL162111 | — | IC50 | = | 48000.0 | nM | 4.32 |