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Assay Detail

CHEMBL662768

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of cell growth was studied in chinese hamster lung cells resistant to actinomycin D (DC-3F/AD-II).
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Cricetulus griseus
Confidence 1 — Organism
Curated By Intermediate

Target

DC3F/AD-II (CHEMBL614283)
Type CELL-LINE
Organism Cricetulus griseus

Publication

Cyclopent[a]anthraquinones as DNA intercalating agents with covalent bond formation potential: synthesis and biological activity.
Kim JY, Su TL, Chou TC, Koehler B, Scarborough A, Ouerfelli O, Watanabe KA.
J Med Chem (1996) 39 : 2812 -2818
PubMed 8709111 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.20 6.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL105 MITOMYCIN 4.0 1 6.96
CHEMBL94680 1 5.44

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL105 MITOMYCIN IC50 = 110.0 nM 6.96
CHEMBL94680 IC50 = 3600.0 nM 5.44